K-252a (from Nonomuraea longicatena chiba) ≥98% (by HPLC)

Supplier: 0000027161

Synonyms: Methyl-6-hydroxy-5-methyl-13-oxo-5,6,7,8,14,15-hexahydro-13h-5,8-epoxy-4b,8a,14-triazadibenzo[b,h]cycloocta[1,2,3,4-jkl]cyclopenta[e]-as-indacene-6-carboxylate

AG-CN2-0019-C100 AG-CN2-0019-M001

102515-726EA 83.08 USD

102515-726 102515-728

K-252a (from Nonomuraea longicatena chiba) ≥98% (by HPLC)

K-252a

K-252a is an antibiotic, PKC, PKA and PKG inhibitor.

Highly potent cell permeable CaM kinase and phosphorylase inhibitor
Apoptosis inducer
Potential drug for psoriasis treatment

Antibiotic. PKC, PKA and PKG inhibitor. Shows neurotropic activity by inducing neurite outgrowth. Tyrosine protein kinase inhibitor of the TRK family. Antiproliferative. Cell cycle arrest inducer.

White to off-white powder

Soluble in DMSO, methanol, methylene chloride, ethyl acetate or acetone. Insoluble in water.

Formula: C₂₇H₂₁N₃O₅
Storage Temperature: Freezer

MDL Number: MFCD00161522
CAS Number: 97161-97-2

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